BAD Molecule Filter
A free machine learning tool by Abdallah Abou Hajal that predicts whether a small molecule will clump into a colloidal aggregate and show up as a false positive in a drug screen.
What it checks
Colloidal aggregation
Give it a molecule as a SMILES string. It predicts whether the molecule is likely to form colloidal aggregates, which inhibit proteins nonspecifically and produce false hits in high-throughput screening. It was Abdallah's MSc work at Al Ain University.
What it does not check
Aggregation only. It does not flag PAINS substructures or other kinds of assay interference, such as reactive or redox cycling compounds.
Run it
Desktop app for Windows and Linux
Version 1.1, free, from the releases page on GitHub.
Source code
Open under the GPL 3.0 licence.
Cite it
Boosting the Accuracy and Chemical Space Coverage of the Detection of Small Colloidal Aggregating Molecules Using the BAD Molecule Filter
Abou Hajal A, Bryce RA, Ben Amor B, Atatreh N, Ghattas MA. Journal of Chemical Information and Modeling 2024, 64(13), 4991-5005.
Cited by
Exploiting colloidal drug aggregation for drug delivery: From promise to prediction using computational tools
Mitigating Molecular Aggregation in Drug Discovery With Predictive Insights From Explainable AI
From Algorithms to Assets: A Comprehensive Review of AI's Role in Preclinical Drug Discovery and the Hurdles to Clinical Translation
For questions about the tool, email Abdallah.